SCHEMBL30723307

SCHEMBL30723307

CCOC(=O)C(CC1CCn2c1nc1c(F)cccc1c2=O)C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.44
HRH3 Q9Y5N1 3/20 0.37
KCNH2 Q12809 2/20 0.37
ADRA1A P35348 1/20 0.37
HTR2C P28335 2/20 0.37
HTR7 P34969 2/20 0.37
HTR2B P41595 2/20 0.37
HTR3A P46098 2/20 0.37
HTR4 Q13639 2/20 0.37
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
HTR1A P08908 1/20 0.35
KDM4E B2RXH2 2/20 0.35
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PDE7A Q13946 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30723324 0.90 KDM4E (0.38) HRH3KCNH2ADRA1AMAPTL3MBTL1
SCHEMBL30723309 0.89 MAPK1 (0.39) TRPV4HRH3KCNH2MAPTL3MBTL1
SCHEMBL30723305 0.88 MAPT (0.40) HRH3KCNH2ADRA1AHTR2CHTR7
SCHEMBL30723322 0.88 MAPT (0.36) TRPV4MAPTL3MBTL1BCHEACHE
SCHEMBL30723313 0.87 CYP1A1 (0.43) HRH3KCNH2HTR7HTR2BHTR4
SCHEMBL30723336 0.84 HRH3 (0.37) HRH3KCNH2BCHEACHEKDM4E
SCHEMBL30723331 0.84 KMT2A (0.34) MAPTL3MBTL1BCHEACHEKDM4E
SCHEMBL30723314 0.84 ACHE (0.54) MAPTL3MBTL1BCHEACHEKDM4E
SCHEMBL30723337 0.82 KMT2A (0.36) HRH3BCHEACHEKDM4ESMN1; SMN2
SCHEMBL30723308 0.80 GAA (0.39) TRPV4HRH3KCNH2HTR7HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117486887-A Polycyclic pyrimidine-4-ketone compound and preparation method and application thereof 昆明学院 2024-02-02 CN disclosed