SCHEMBL30723456

SCHEMBL30723456

CC(C)(C)OC(=O)N1C[C@@H](OC(=O)c2ccccc2)[C@H]2[C@@H]1CN2Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KLK7 P49862 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30723543 1.00 PDK1 (0.40) PDK1PDK2PDK3PDK4HDAC1
SCHEMBL30892168 0.83 NR1H2 (0.42) PDK1PDK2PDK3PDK4KLK7
SCHEMBL30723476 0.83 NR1H2 (0.42) PDK1PDK2PDK3PDK4KLK7
SCHEMBL30723469 0.82 MAPT (0.44) PDK1PDK2PDK3PDK4JAK2
SCHEMBL30723442 0.82 MAPT (0.44) PDK1PDK2PDK3PDK4JAK2
SCHEMBL30723461 0.81 PDK1 (0.41) PDK1PDK2PDK3PDK4KLK7
SCHEMBL30723486 0.81 ABCB1 (0.41) PDK1PDK2PDK3PDK4CHRM2
SCHEMBL30723440 0.80 SIRT1 (0.41) PDK1PDK2PDK3PDK4KLK7
SCHEMBL30723511 0.79 KMT2A (0.40) PDK1PDK2PDK3PDK4CHRM2
SCHEMBL30723528 0.79 KMT2A (0.40) PDK1PDK2PDK3PDK4CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118027068-A Compound containing bridged ring and application thereof 上海艾力斯医药科技股份有限公司 2024-05-14 CN disclosed
CN-117430619-A Pyrazolopyridine compound and preparation method and application thereof 上海艾力斯医药科技股份有限公司 2024-01-23 CN disclosed