SCHEMBL30725866

SCHEMBL30725866

N#Cc1ccc(C(=O)Nc2ccc3[nH]nc(-c4cccnc4)c3c2)cc1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 17/20 0.70
ITK Q08881 1/20 0.60
CYP11B1 P15538 1/20 0.60
CYP11B2 P19099 1/20 0.60
ABL1 P00519 1/20 0.56
PDGFRB P09619 1/20 0.56
BCR P11274 1/20 0.56
PDGFRA P16234 1/20 0.56
PRKCA P17252 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29172510 1.00 LRRK2 (0.70) LRRK2ITKCYP11B1CYP11B2ABL1
SCHEMBL29172536 0.90 LRRK2 (0.68) LRRK2
SCHEMBL30725856 0.90 LRRK2 (0.68) LRRK2
SCHEMBL30725877 0.87 CDK7 (0.67) LRRK2ITK
SCHEMBL29172495 0.87 CDK7 (0.67) LRRK2ITK
SCHEMBL30725869 0.86 LRRK2 (0.58) LRRK2ITK
SCHEMBL30725858 0.86 DYRK1A (0.61) LRRK2ITKCYP11B1CYP11B2ABL1
SCHEMBL29172502 0.86 DYRK1A (0.61) LRRK2ITKCYP11B1CYP11B2ABL1
SCHEMBL29172497 0.86 LRRK2 (0.58) LRRK2ITK
SCHEMBL22890022 0.83 LRRK2 (1.00) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186066-A Indazole ALK5 inhibitor and preparation method and application thereof 中国药科大学 2023-12-08 CN disclosed