SCHEMBL30725867

SCHEMBL30725867

C[Si](C)(C)CCOCn1nc(-c2cccnc2)c2cc(NC(=O)c3cccc(F)c3)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.45
CSF1R P07333 1/20 0.43
GSK3B P49841 1/20 0.43
ABL1 P00519 3/20 0.40
BCR P11274 3/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ROCK2 O75116 2/20 0.40
TEK Q02763 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
TP53 P04637 1/20 0.39
ALDH1A1 P00352 1/20 0.39
NAMPT P43490 1/20 0.38
EPHX2 P34913 1/20 0.38
PDPK1 O15530 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29172485 1.00 BRAF (0.45) BRAFCSF1RGSK3BABL1BCR
SCHEMBL29172517 0.92 CYP11B1 (0.47) ABL1BCRMAPTKDM4EABCG2
SCHEMBL30725853 0.92 CYP11B1 (0.47) ABL1BCRMAPTKDM4EABCG2
SCHEMBL29172524 0.91 PRKCA (0.43) ABL1BCRMAPTNPC1RAB9A
SCHEMBL30725845 0.89 BRAF (0.48) BRAFABL1BCRMAPTKDM4E
SCHEMBL29172518 0.89 BRAF (0.48) BRAFABL1BCRMAPTKDM4E
SCHEMBL30725863 0.87 MAPT (0.47) MAPTKDM4ETEKNPC1RAB9A
SCHEMBL29172525 0.87 MAPT (0.47) MAPTKDM4ETEKNPC1RAB9A
SCHEMBL30725850 0.85 L3MBTL1 (0.46) MAPTKDM4ENPC1RAB9AALDH1A1
SCHEMBL30725852 0.85 CYP11B1 (0.46) BRAFABL1BCRMAPTROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186066-A Indazole ALK5 inhibitor and preparation method and application thereof 中国药科大学 2023-12-08 CN disclosed