SCHEMBL30726153

SCHEMBL30726153

CC(Cc1cc(F)cc(C(N)=O)c1F)N(C)C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP14 Q460N5 3/20 0.37
HTR2A P28223 1/20 0.36
RIPK1 Q13546 4/20 0.35
PARP1 P09874 4/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DPP4 P27487 1/20 0.33
DPP9 Q86TI2 1/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
P4HB P07237 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30726152 0.79 P4HB (0.40) HTR2APARP1P4HBMEN1KMT2A
SCHEMBL30726149 0.72 P4HB (0.47) HTR2ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL24455315 0.69 CES2 (0.45) PARP14PARP1CES2CES1
SCHEMBL6186161 0.67 PARP1 (0.41) PARP14PARP1CES2CES1
SCHEMBL10160070 0.67 POLB (0.45) PARP1POLBL3MBTL1CES2CES1
SCHEMBL477698 0.66 CES2 (0.68) PARP1CES2CES1
SCHEMBL15094272 0.65 KCNJ6 (0.36) PARP1CES2CES1
SCHEMBL29088228 0.63 PARP1 (0.43) PARP1CES2CES1MEN1KMT2A
SCHEMBL29851114 0.63 PARP1 (0.43) PARP1CES2CES1MEN1KMT2A
SCHEMBL22169000 0.63 PARP1 (0.40) PARP14PARP1L3MBTL1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117425644-A Opioid receptor modulators 埃皮欧黛公司 2024-01-19 CN disclosed