SCHEMBL30728638

SCHEMBL30728638

O=C1CCc2cc(OCCCCN3CCN(Cc4ccccc4)CC3)cc3c2N1CC3

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.58
MAOB P27338 4/20 0.58
ACHE P22303 2/20 0.52
CHRM2 P08172 1/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51
CHRM1 P11229 1/20 0.51
DRD2 P14416 1/20 0.51
CHRM3 P20309 1/20 0.51
DRD4 P21917 1/20 0.51
DRD3 P35462 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23409228 1.00 MAOA (0.58) MAOAMAOBACHECHRM2CHRM4
SCHEMBL23409234 0.83 LMNA (0.49) CHRM1DRD2DRD3
SCHEMBL23409205 0.82 DRD3 (0.62) MAOAMAOBDRD2DRD4DRD3
SCHEMBL23409975 0.81 DRD2 (0.53) DRD2DRD4DRD3
SCHEMBL23409561 0.81 HRH3 (0.46) MAOAMAOB
SCHEMBL23409211 0.81 DRD2 (0.53) MAOBDRD2DRD4DRD3
SCHEMBL23409236 0.80 DRD2 (0.62) MAOAMAOBACHECHRM2CHRM1
SCHEMBL30728639 0.80 DRD2 (0.62) MAOAMAOBACHECHRM2CHRM1
SCHEMBL30728641 0.77 DRD2 (0.67) DRD2
SCHEMBL23409242 0.77 DRD2 (0.61) MAOAMAOBACHECHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728956-B Fused heterocyclic derivative and application thereof 上海枢境生物科技有限公司 2024-01-12 CN disclosed