SCHEMBL30730839

SCHEMBL30730839

COC(=O)c1cc2c(-c3cnc(N)c(-c4ccc(N5CCCC5=O)cc4)c3)ccnc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 2/20 0.41
DGAT2 Q96PD7 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 2/20 0.38
HTT P42858 1/20 0.38
NUDT1 P36639 1/20 0.38
TGFBR1 P36897 2/20 0.38
PRKAB2 O43741 1/20 0.38
PRKAG1 P54619 1/20 0.38
PRKAA2 P54646 1/20 0.38
PRKAA1 Q13131 1/20 0.38
PRKAG3 Q9UGI9 1/20 0.38
PRKAG2 Q9UGJ0 1/20 0.38
PRKAB1 Q9Y478 1/20 0.38
MAP4K4 O95819 1/20 0.37
PDGFRB P09619 1/20 0.36
KDR P35968 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22553751 1.00 TBK1 (0.41) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL22553938 0.88 NUDT1 (0.43) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL30730826 0.88 NUDT1 (0.43) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL30731117 0.88 NUDT1 (0.43) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL22554042 0.85 DGAT2 (0.40) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL30730806 0.85 DGAT2 (0.40) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL22553861 0.82 NUDT1 (0.41) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL30777590 0.82 NUDT1 (0.41) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL22554168 0.82 NUDT1 (0.41) TBK1DGAT2SMN1; SMN2MAPTNPC1
SCHEMBL30730817 0.82 NUDT1 (0.41) TBK1DGAT2SMN1; SMN2MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN claimed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed