SCHEMBL30734232

SCHEMBL30734232

Nc1cc(-c2ccc3ncnc(N4CCN(c5ccc(O)cc5)CC4)c3c2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.49
MEN1 O00255 7/20 0.49
KMT2A Q03164 7/20 0.49
KDM4E B2RXH2 3/20 0.49
MAPT P10636 2/20 0.49
GAA P10253 1/20 0.49
MCL1 Q07820 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CYP3A4 P08684 15/20 0.49
CLK4 Q9HAZ1 13/20 0.49
CYP1A2 P05177 13/20 0.49
HIF1A Q16665 10/20 0.49
LMNA P02545 9/20 0.49
MAPK1 P28482 9/20 0.49
CYP2D6 P10635 10/20 0.48
USP2 O75604 8/20 0.48
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30734233 0.89 ACHE (0.55) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL30734231 0.89 CYP3A4 (0.52) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL30734187 0.89 ACHE (0.53) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL30734169 0.83 CYP3A4 (0.54) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL30734142 0.83 MAP4K4 (0.44) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL30734171 0.83 CYP1A2 (0.62) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL30734129 0.81 ACHE (0.55) ALDH1A1MEN1KMT2AKDM4ECYP3A4
SCHEMBL30734206 0.80 CYP3A4 (0.50) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL30734203 0.80 ACHE (0.56) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL31745183 0.79 MEN1 (0.54) ALDH1A1MEN1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250382301-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF UNIV ARIZONA (US) 2025-12-18 US disclosed
EP-4543888-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF Arizona Board of Regents on behalf of The University of Arizona (US) 2025-04-30 EP disclosed
WO-2023250083-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2023-12-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250382301-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF CLK2, CLK3, CLK1 ALDH1A1 4568/4885MEN1 407/4885KMT2A 2060/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.