SCHEMBL3073564

SCHEMBL3073564

CN(Cc1ccccc1)Cc1coc(-c2ccc(OCCCN3CCCCC3)cc2)n1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.67
BCHE P06276 5/20 0.60
ACHE P22303 5/20 0.60
KCNH2 Q12809 3/20 0.53
HRH1 P35367 1/20 0.53
TLR9 Q9NR96 1/20 0.51
ATP4A P20648 2/20 0.49
ATP4B P51164 2/20 0.49
HRH4 Q9H3N8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3085069 0.84 HRH3 (0.66) HRH3KCNH2TLR9
SCHEMBL3569235 0.82 BCHE (0.83) HRH3BCHEACHEKCNH2HRH1
SCHEMBL3081656 0.81 HRH3 (1.00) HRH3ACHEKCNH2HRH1TLR9
SCHEMBL3070984 0.81 HRH3 (1.00) HRH3ACHEKCNH2HRH1TLR9
SCHEMBL3082345 0.81 HRH3 (1.00) HRH3ACHEKCNH2HRH1TLR9
SCHEMBL3072910 0.80 HRH3 (0.81) HRH3KCNH2HRH1TLR9
SCHEMBL3061479 0.79 HRH3 (0.98) HRH3ACHEKCNH2HRH1TLR9
SCHEMBL16523574 0.78 ACHE (0.66) HRH3BCHEACHEHRH1
SCHEMBL3081190 0.76 HRH3 (0.84) HRH3ACHEKCNH2HRH1TLR9
SCHEMBL3072689 0.76 HRH3 (0.80) HRH3KCNH2HRH1TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790720-B2 Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses UCB PHARMA, S.A. (BE) 2010-09-07 US claimed
US-20080275046-A1 Compounds Comprising an Oxazole or Thiazole Moiety, Processes for Making Them, and Their Uses UCB PHARMA, S.A. (BE) 2008-11-06 US claimed
EP-1866293-A1 COMPOUNDS COMPRISING AN OXAZOLE OR THIAZOLE MOIETY, PROCESSES FOR MAKING THEM, AND THEIR USES UCB Pharma, S.A. (BE) 2007-12-19 EP claimed
WO-2006103045-A1 COMPOUNDS COMPRISING AN OXAZOLE OR THIAZOLE MOIETY, PROCESSES FOR MAKING THEM, AND THEIR USES UCB PHARMA S.A. (BE) 2006-10-05 WO claimed
US-7790720-B2 Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses UCB PHARMA, S.A. (BE) 2010-09-07 US disclosed
US-20080275046-A1 Compounds Comprising an Oxazole or Thiazole Moiety, Processes for Making Them, and Their Uses UCB PHARMA, S.A. (BE) 2008-11-06 US disclosed
EP-1866293-A1 COMPOUNDS COMPRISING AN OXAZOLE OR THIAZOLE MOIETY, PROCESSES FOR MAKING THEM, AND THEIR USES UCB Pharma, S.A. (BE) 2007-12-19 EP disclosed
WO-2006103045-A1 COMPOUNDS COMPRISING AN OXAZOLE OR THIAZOLE MOIETY, PROCESSES FOR MAKING THEM, AND THEIR USES UCB PHARMA S.A. (BE) 2006-10-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080275046-A1 Compounds Comprising an Oxazole or Thiazole Moiety, Processes for Making Them, and Their Uses OXER1, OXTR, OGFR HRH3 4/4885BCHE 1536/4885ACHE 1842/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.