SCHEMBL3073945

SCHEMBL3073945

CN1CCC(Oc2ccccc2F)c2ccc(N3C=CC=CC3)cc2C1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
KMT2A Q03164 1/20 0.31
MAPT P10636 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
MAP4K1 Q92918 1/20 0.31
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3083318 0.89 MCHR1 (0.37) SSTR4SLC6A4MAPTESR2HTR2C
SCHEMBL3081797 0.87 ESR1 (0.35) SSTR4SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL3094904 0.82 MCHR1 (0.38) SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL3477654 0.79 SSTR4 (0.36) SSTR4SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL3093435 0.75 SSTR4 (0.37) SSTR4SLC6A2SLC6A4SLC6A3KMT2A
SCHEMBL3099039 0.74 SLC6A4 (0.47) SSTR4SLC6A2SLC6A4SLC6A3MAP4K1
SCHEMBL3086267 0.73 GSK3B (0.41) SSTR4SLC6A2SLC6A4SLC6A3MAP4K1
SCHEMBL3087454 0.72 ROCK2 (0.43) MAP4K1
SCHEMBL3079430 0.72 HTR2C (0.39) SSTR4SLC6A4HTR2C
SCHEMBL3476770 0.72 NOS1 (0.42) SSTR4SLC6A2SLC6A4SLC6A3MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2146720-A1 ARYLOXY-AND HETEROARYLOXY-SUBSTITUTED TETRAHYDROBENZAZEPINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR Technology, Inc. (US) 2010-01-27 EP disclosed
WO-2008141082-A1 ARYLOXY-AND HETEROARYLOXY-SUBSTITUTED TETRAHYDROBENZAZEPINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR TECHNOLOGY, INC. (US) 2008-11-20 WO disclosed