SCHEMBL30740717

SCHEMBL30740717

COc1cccc2c(C(C)N)c[nH]c12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.54
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 2/20 0.48
HPGD P15428 2/20 0.48
HTR6 P50406 1/20 0.48
DYRK1A Q13627 2/20 0.46
NFATC1 O95644 1/20 0.46
GSK3B P49841 1/20 0.46
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19040093 0.87 HTR2A (0.53) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL31000552 0.81 ALDH1A1 (0.52) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL30024944 0.79 ALDH1A1 (0.57) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL7870399 0.78 SOS2 (0.68) HTR2AHTR6MTNR1AMTNR1BSOS2
SCHEMBL31037788 0.76 HDAC3 (0.56) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL8926562 0.74 HTR2A (0.57) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL17187807 0.74 IDO1 (0.46) HDAC4HDAC8ALDH1A1MEN1LMNA
SCHEMBL10466658 0.74 HDAC3 (0.46) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL8926558 0.73 HTR2A (0.55) HTR2AHDAC3HDAC4HDAC1HDAC7
SCHEMBL20673987 0.73 KDM4E (0.56) HTR2AHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117043154-A GPCR receptor agonists, pharmaceutical compositions comprising same, and methods of use thereof 卡莫特医疗有限公司 2023-11-10 CN disclosed