SCHEMBL30745481

SCHEMBL30745481

COc1ccc(C(=O)/C=C/c2ccc(Cl)cc2)c(O)c1CNCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.53
HDAC3 O15379 3/20 0.53
HDAC1 Q13547 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC8 Q9BY41 3/20 0.53
MEN1 O00255 1/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 1/20 0.53
KMT2A Q03164 1/20 0.53
ABCG2 Q9UNQ0 5/20 0.50
CYP1A1 P04798 2/20 0.49
CYP1B1 Q16678 2/20 0.49
CYP1A2 P05177 1/20 0.49
APP P05067 2/20 0.48
AR P10275 1/20 0.46
MAOA P21397 1/20 0.46
ABCB1 P08183 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745460 0.91 HDAC3 (0.53) MAOBHDAC3HDAC1HDAC2HDAC8
SCHEMBL30745477 0.90 HDAC3 (0.55) MAOBHDAC3HDAC1HDAC2HDAC8
SCHEMBL30745452 0.88 MEN1 (0.52) MAOBHDAC3HDAC1HDAC2HDAC8
SCHEMBL30745475 0.81 ABCG2 (0.52) MAOBHDAC3HDAC1HDAC2HDAC8
SCHEMBL30745438 0.79 MAOB (0.58) MAOBMEN1LMNAMAPTKMT2A
SCHEMBL5517453 0.79 MAOB (0.67) MAOBMEN1LMNAMAPTKMT2A
SCHEMBL5517451 0.79 MAOB (0.67) MAOBMEN1LMNAMAPTKMT2A
SCHEMBL30745478 0.77 MAOB (0.56) MAOBMEN1LMNAMAPTKMT2A
SCHEMBL30745498 0.75 MAOB (0.53) MAOBMEN1LMNAMAPTKMT2A
SCHEMBL30745496 0.74 MAOB (0.53) MAOBMEN1LMNAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN claimed
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN disclosed