SCHEMBL30745475

SCHEMBL30745475

COc1cc(O)c(C(=O)/C=C/c2ccc(Cl)cc2)cc1CNCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.52
MAOB P27338 1/20 0.52
APP P05067 2/20 0.52
AR P10275 3/20 0.51
HDAC3 O15379 3/20 0.51
HDAC1 Q13547 3/20 0.51
HDAC2 Q92769 3/20 0.51
HDAC8 Q9BY41 3/20 0.51
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
CXCL12 P48061 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745479 0.91 APP (0.52) ABCG2APPHDAC3HDAC1HDAC2
SCHEMBL30745447 0.90 ACHE (0.60) ABCG2MAOBAPPARHDAC3
SCHEMBL30745466 0.89 MAOA (0.53) MAOBAPPHDAC3HDAC1HDAC2
SCHEMBL30745510 0.85 ABCG2 (0.53) ABCG2MAOBARACHEBACE1
SCHEMBL30745481 0.81 MAOB (0.53) ABCG2MAOBAPPARHDAC3
SCHEMBL25228491 0.79 AR (0.70) ABCG2MAOBARACHEBACE1
SCHEMBL30745470 0.79 AR (0.58) ABCG2MAOBARACHEBACE1
SCHEMBL30745458 0.79 AR (0.57) ABCG2MAOBARACHEBACE1
SCHEMBL30745511 0.75 SMN1; SMN2 (0.53) ABCG2MAOBAPPARACHE
SCHEMBL5088647 0.75 MAPT (0.62) ABCG2ARACHEBACE1CXCL12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN claimed
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN disclosed