SCHEMBL30745477

SCHEMBL30745477

COc1ccc(C(=O)/C=C/c2ccc(F)cc2)c(O)c1CNCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.55
HDAC1 Q13547 3/20 0.55
HDAC2 Q92769 3/20 0.55
HDAC8 Q9BY41 3/20 0.55
CTSL P07711 2/20 0.53
MAOB P27338 4/20 0.53
MEN1 O00255 1/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 1/20 0.53
KMT2A Q03164 1/20 0.53
CYP1B1 Q16678 2/20 0.49
CYP1A1 P04798 1/20 0.49
CYP1A2 P05177 1/20 0.49
ABCG2 Q9UNQ0 2/20 0.49
TUBB4A P04350 1/20 0.48
TUBB P07437 1/20 0.48
TUBA3C P0DPH7 1/20 0.48
TUBA1B P68363 1/20 0.48
TUBA4A P68366 1/20 0.48
TUBB4B P68371 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745460 0.91 HDAC3 (0.53) HDAC3HDAC1HDAC2HDAC8MAOB
SCHEMBL30745481 0.90 MAOB (0.53) HDAC3HDAC1HDAC2HDAC8MAOB
SCHEMBL30745452 0.88 MEN1 (0.52) HDAC3HDAC1HDAC2HDAC8MAOB
SCHEMBL30745447 0.81 ACHE (0.60) HDAC3HDAC1HDAC2HDAC8CTSL
SCHEMBL30745507 0.79 CTSL (0.59) CTSLMAOBMEN1LMNAMAPT
SCHEMBL5517451 0.79 MAOB (0.67) CTSLMAOBMEN1LMNAMAPT
SCHEMBL5517453 0.79 MAOB (0.67) CTSLMAOBMEN1LMNAMAPT
SCHEMBL30745464 0.77 CTSL (0.57) CTSLMAOBMEN1LMNAMAPT
SCHEMBL30745465 0.75 CTSL (0.54) CTSLMAOBMEN1LMNAMAPT
SCHEMBL30745473 0.74 CTSL (0.53) CTSLMAOBMEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN claimed
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN disclosed