SCHEMBL30765382

SCHEMBL30765382

O=C(O)c1ccc(-c2cc3nccc(Cl)c3o2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 7/20 0.48
RARB P10826 7/20 0.48
RARG P13631 7/20 0.48
KMO O15229 2/20 0.43
MAPKAPK2 P49137 1/20 0.42
TNKS O95271 1/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30765288 0.88 MAPT (0.39) RARARARBRARGKDM4ENPC1
SCHEMBL18339379 0.84 CYP1A2 (0.40) RARARARBRARGKDM4ETDP1
SCHEMBL30765301 0.84 TNKS (0.45) TNKSKDM4ETDP1NPC1RAB9A
SCHEMBL18339400 0.84 TNKS (0.45) TNKSKDM4ETDP1NPC1RAB9A
SCHEMBL15209535 0.83 RARA (0.39) RARARARBRARGKMORXRA
SCHEMBL722060 0.82 CYP1A1 (0.47) TNKSKDM4ENPC1RAB9AMEN1
SCHEMBL15173516 0.81 RAB9A (0.48) RARARARBRARGTNKSKDM4E
SCHEMBL723467 0.81 HPGD (0.48) NPC1RAB9AMEN1ALDH1A1MAPT
SCHEMBL721875 0.80 CSNK2A2 (0.40) MAPKAPK2TNKSKDM4ENPC1RAB9A
SCHEMBL724007 0.80 MAPK14 (0.43) TNKSKDM4ENPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024033280-A1 FUROPYRIDIN AND FUROPYRIMIDIN, INHIBITORS OF PI4K, FOR USE IN THE TREATMENT OF PARASITE INFECTION AND MALARIA MERCK PATENT GMBH (DE) 2024-02-15 WO disclosed