SCHEMBL30767660

SCHEMBL30767660

CC(F)(F)c1ccc(-c2ccc(CO)cc2)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.47
FYN P06241 5/20 0.42
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
KIF11 P52732 2/20 0.40
GCK P35557 1/20 0.40
GCKR Q14397 1/20 0.40
BRS3 P32247 2/20 0.39
KCNH2 Q12809 2/20 0.39
MAPT P10636 1/20 0.38
STAT3 P40763 1/20 0.38
ATM Q13315 1/20 0.38
TP53 P04637 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
PPARA Q07869 1/20 0.38
MAOB P27338 1/20 0.38
SLC22A12 Q96S37 1/20 0.37
GRM2 Q14416 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2269528 0.87 KIF11 (0.51) KDM1AFYNKIF11GCKGCKR
SCHEMBL31375486 0.84 RAB9A (0.40) KDM1ANPC1RAB9ASMN1; SMN2KIF11
SCHEMBL30767444 0.84 KIF11 (0.40) KDM1ANPC1RAB9ASMN1; SMN2KIF11
SCHEMBL30633001 0.81 PPARA (0.50) KDM1AFYNNPC1RAB9ASMN1; SMN2
SCHEMBL1549725 0.81 PPARA (0.50) KDM1AFYNNPC1RAB9ASMN1; SMN2
SCHEMBL31375576 0.80 KDM1A (0.44) KDM1AKIF11GCKGCKRBRS3
SCHEMBL1742369 0.77 EPHX2 (0.44) KIF11PPARA
SCHEMBL21034957 0.75 KDM1A (0.47) KDM1AFYNNPC1RAB9ASMN1; SMN2
SCHEMBL17954213 0.75 SMN1; SMN2 (0.66) KDM1AFYNNPC1RAB9ASMN1; SMN2
SCHEMBL508027 0.75 FYN (0.56) KDM1AFYNNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4568960-A1 BICYCLIC TETRAHYDROAZEPINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2025-06-18 EP disclosed
WO-2024033458-A1 BICYCLIC TETRAHYDROAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2024-02-15 WO disclosed