SCHEMBL30775557

SCHEMBL30775557

Nc1ncnc2ccc(Br)c(F)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 15/20 0.40
PI4KA P42356 1/20 0.37
PI4K2B Q8TCG2 1/20 0.37
PI4K2A Q9BTU6 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
TDP2 O95551 1/20 0.35
NSD2 O96028 1/20 0.35
PAX8 Q06710 1/20 0.35
HKDC1 Q2TB90 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
MINK1 Q8N4C8 1/20 0.35
TNIK Q9UKE5 1/20 0.35
PIK3CD O00329 1/20 0.34
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
HCK P08631 1/20 0.34
SRC P12931 1/20 0.34
KDR P35968 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29936178 0.78 PDE4A (0.37) EGFRKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL17665817 0.78 LIMK1 (0.41) MAP4K4PI4KAPI4K2BPI4K2API4KB
SCHEMBL25167004 0.74 DHFR (0.42)
SCHEMBL30770136 0.74 TDP2 (0.45) MAP4K4PI4KBTDP2NSD2PAX8
SCHEMBL30097809 0.74 TDP2 (0.45) MAP4K4PI4KBTDP2NSD2PAX8
SCHEMBL18312022 0.73 PI4KA (0.48) MAP4K4PI4KAPI4K2BPI4K2API4KB
SCHEMBL29129392 0.70 CSNK2A1 (0.38) MAP4K4MINK1TNIKEPHB4
SCHEMBL31728512 0.70 MAP4K4 (0.37) MAP4K4PI4KAPI4K2BPI4K2API4KB
SCHEMBL2124702 0.69 PI4KA (0.48) MAP4K4PI4KAPI4K2BPI4K2API4KB
SCHEMBL18420628 0.67 CCNB2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117500803-A Amino-substituted heterocycles for the treatment of cancers with EGFR mutations 纽威伦特公司 2024-02-02 CN disclosed