SCHEMBL30775559

SCHEMBL30775559

Nc1c(F)cnc2ccc(Cl)nc12

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.35
EGFR P00533 1/20 0.32
PIK3CA P42336 1/20 0.31
BACE1 P56817 1/20 0.31
MAPT P10636 1/20 0.31
MAP4K4 O95819 2/20 0.31
MELK Q14680 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21494203 0.81 EGFR (0.33) EGFRMELK
SCHEMBL23020432 0.75 KCNH2 (0.34) EGFRMELK
SCHEMBL3379185 0.75 MAP4K4 (0.41) PIK3CDEGFRPIK3CAMAPTMAP4K4
SCHEMBL30775555 0.75 MAP4K4 (0.41) PIK3CDEGFRPIK3CAMAPTMAP4K4
SCHEMBL16748191 0.72 MAPT (0.40) MAPT
SCHEMBL9955167 0.70 ALDH1A1 (0.41) PIK3CA
SCHEMBL29439641 0.68 MAP4K4 (0.54) MAP4K4
SCHEMBL22715644 0.68 NR4A2 (0.47) PIK3CDEGFRMAPT
SCHEMBL15587364 0.68 MAP4K4 (0.54) MAP4K4
SCHEMBL21914082 0.68 PIK3CD (0.33) PIK3CDEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117500803-A Amino-substituted heterocycles for the treatment of cancers with EGFR mutations 纽威伦特公司 2024-02-02 CN disclosed