SCHEMBL30779221

SCHEMBL30779221

CC(C)(C)OC(=O)NCc1cccc(NC2CCCC2)c1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.54
BRD4 O60885 3/20 0.48
JAK2 O60674 1/20 0.47
JAK1 P23458 1/20 0.47
CREBBP Q92793 1/20 0.46
GLS O94925 3/20 0.44
EPHX1 P07099 1/20 0.44
NAMPT P43490 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
USP30 Q70CQ3 1/20 0.43
CCKBR P32239 1/20 0.43
CYP3A4 P08684 1/20 0.43
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24732888 1.00 ROCK2 (0.54) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL15348038 0.85 ALDH1A1 (0.46) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL15348037 0.85 ALDH1A1 (0.46) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL13334315 0.82 BCHE (0.45) ROCK2BRD4
SCHEMBL31709823 0.81 BRD4 (0.54) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL731764 0.81 BRD4 (0.54) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL25048390 0.81 BRD4 (0.47) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL7238726 0.80 BRD4 (0.48) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL14894253 0.79 JAK2 (0.45) ROCK2BRD4JAK2JAK1CREBBP
SCHEMBL20246342 0.79 JAK2 (0.49) ROCK2BRD4JAK2JAK1CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805341-B Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2023-12-08 CN disclosed