SCHEMBL30786158

SCHEMBL30786158

CNC(=O)c1cc(F)ccc1Sc1ccc2c(/C=C/c3cnn(CCCN4CCCC4)c3)nn(C3CCCCO3)c2c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.34
HTR2A P28223 8/20 0.34
HTR1A P08908 4/20 0.34
HTR2C P28335 3/20 0.34
ADRA1A P35348 3/20 0.34
HRH1 P35367 3/20 0.34
KCNH2 Q12809 2/20 0.34
PLK4 O00444 2/20 0.30
AURKA O14965 2/20 0.30
MAP4K4 O95819 2/20 0.30
PAK4 O96013 2/20 0.30
ABL1 P00519 2/20 0.30
LCK P06239 2/20 0.30
CSF1R P07333 2/20 0.30
RET P07949 2/20 0.30
MET P08581 2/20 0.30
PDGFRB P09619 2/20 0.30
KIT P10721 2/20 0.30
FGFR1 P11362 2/20 0.30
PDGFRA P16234 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31475173 0.93 HTR2A (0.35) DRD2HTR2AHTR1AAXLKDR
SCHEMBL30786082 0.89 DRD2 (0.35) DRD2HTR2AHTR1A
SCHEMBL31475169 0.86 CNR1 (0.34) PLK4AURKAMAP4K4PAK4ABL1
SCHEMBL31475199 0.85 KDR (0.34) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL30786126 0.83 DRD2 (0.32) DRD2HTR2AHTR1AAXLMERTK
SCHEMBL31475194 0.80 KDR (0.34) PLK4AURKAMAP4K4PAK4ABL1
SCHEMBL31475185 0.80 KDR (0.34) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL31475210 0.80 DRD2 (0.37) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL30786134 0.79 KDR (0.38) DRD2HTR2AHTR1AHTR2CADRA1A
SCHEMBL30786236 0.79 KDR (0.37) DRD2HTR2AHTR1AKDRBMPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119604488-A Protein tyrosine kinase inhibitor and medical application thereof 苏州必扬医药科技有限公司 2025-03-11 CN disclosed
WO-2024032584-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF 苏州必扬医药科技有限公司 2024-02-15 WO disclosed