SCHEMBL30786126

SCHEMBL30786126

CCNC(=O)c1cccc(F)c1Sc1ccc2c(/C=C/c3cnn(CCCN4CCCC4)c3)nn(C3CCCCO3)c2c1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
SMYD2 Q9NRG4 1/20 0.31
AXL P30530 1/20 0.31
TYRO3 Q06418 1/20 0.31
MERTK Q12866 1/20 0.31
HTR1A P08908 1/20 0.30
CTSS P25774 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31475169 0.90 CNR1 (0.34) CNR1CNR2SMYD2AXLMERTK
SCHEMBL30786082 0.89 DRD2 (0.35) DRD2HTR2ACNR1CNR2HTR1A
SCHEMBL31475216 0.86 DRD2 (0.33) DRD2HTR2AHTR1A
SCHEMBL30786128 0.86 CNR1 (0.31) CNR1CNR2
SCHEMBL30786158 0.83 DRD2 (0.34) DRD2HTR2AAXLMERTKHTR1A
SCHEMBL31475173 0.81 HTR2A (0.35) DRD2HTR2ACNR1CNR2AXL
SCHEMBL30786218 0.81 KDR (0.31)
SCHEMBL30786135 0.79 KDR (0.35) CNR1CNR2
SCHEMBL30786231 0.79 DGAT2 (0.35) CNR1CNR2AXLTYRO3MERTK
SCHEMBL30786078 0.78 KDR (0.36) DRD2HTR2ACNR1CNR2AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119604488-A Protein tyrosine kinase inhibitor and medical application thereof 苏州必扬医药科技有限公司 2025-03-11 CN disclosed
WO-2024032584-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF 苏州必扬医药科技有限公司 2024-02-15 WO disclosed