SCHEMBL30789201

SCHEMBL30789201

NC(=O)Cc1cccc2c1CN(C(=O)c1c(O)cc(O)cc1OCc1ccccc1)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.43
HSP90AB1 P08238 2/20 0.43
TRAP1 Q12931 4/20 0.39
HSP90B1 P14625 2/20 0.39
PTGER1 P34995 2/20 0.38
PTGER4 P35408 2/20 0.38
PTGER3 P43115 2/20 0.38
PTGER2 P43116 2/20 0.38
CFD P00746 2/20 0.37
PLG P00747 1/20 0.37
PLAU P00749 1/20 0.37
F11 P03951 1/20 0.37
KLKB1 P03952 1/20 0.37
F7 P08709 1/20 0.37
TPSB2 P20231 1/20 0.37
SPR P35270 1/20 0.36
FOLH1 Q04609 1/20 0.35
SLC5A1 P13866 1/20 0.35
SLC5A2 P31639 1/20 0.35
RXRB P28702 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29168708 1.00 HSP90AA1 (0.43) HSP90AA1HSP90AB1TRAP1HSP90B1PTGER1
SCHEMBL30156544 0.90 TRAP1 (0.40) HSP90AA1HSP90AB1TRAP1HSP90B1PTGER1
SCHEMBL24913931 0.90 TRAP1 (0.40) HSP90AA1HSP90AB1TRAP1HSP90B1PTGER1
Hydrochloric Acid SCHEMBL30156871 0.90 TRAP1 (0.39) HSP90AA1HSP90AB1TRAP1HSP90B1PTGER1
SCHEMBL24913845 0.86 TRAP1 (0.41) HSP90AA1HSP90AB1TRAP1HSP90B1SPR
SCHEMBL30156653 0.86 TRAP1 (0.41) HSP90AA1HSP90AB1TRAP1HSP90B1SPR
SCHEMBL24913814 0.86 HSP90AB1 (0.45) HSP90AA1HSP90AB1TRAP1HSP90B1PTGER1
SCHEMBL30155911 0.86 HSP90AB1 (0.45) HSP90AA1HSP90AB1TRAP1HSP90B1PTGER1
SCHEMBL24913881 0.85 TRAP1 (0.51) HSP90AA1HSP90AB1TRAP1HSP90B1SPR
SCHEMBL30156809 0.85 TRAP1 (0.51) HSP90AA1HSP90AB1TRAP1HSP90B1SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117693507-A Inhibitor compounds 奈奥芬莱有限公司 2024-03-12 CN disclosed