SCHEMBL30832011

SCHEMBL30832011

COc1ncccc1CNC(=O)N(C)CC1CCN(CC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
CHRM4 P08173 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HTR2A P28223 2/20 0.40
HTR1A P08908 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
HTR2C P28335 1/20 0.39
KCNH2 Q12809 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29208020 0.95 CHRM4 (0.41) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL30832001 0.90 ALDH1A1 (0.47) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
Trifluoroacetic Acid SCHEMBL29207970 0.85 ALDH1A1 (0.43) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL30832006 0.83 KDM4E (0.47) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL30832047 0.82 TSHR (0.47) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL29208106 0.82 HTR2A (0.51) HTTSMN1; SMN2CHRM4KMT2AHTR2A
SCHEMBL30832045 0.81 LMNA (0.52) ALDH1A1TSHRKDM4ESMN1; SMN2KMT2A
SCHEMBL30831993 0.80 MMP13 (0.42) ALDH1A1TSHRKDM4EHTR2AHTR2C
SCHEMBL30832023 0.80 MLLT1 (0.43) ALDH1A1TSHRKDM4EHTTSMN1; SMN2
SCHEMBL30832048 0.80 KIT (0.43) ALDH1A1TSHRKDM4EHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed