SCHEMBL30832013

SCHEMBL30832013

CC(C)(C)OC(=O)NCC1CCN(CC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.49
HTR2A P28223 4/20 0.47
HTR2C P28335 3/20 0.47
KCNH2 Q12809 3/20 0.47
HTR2B P41595 2/20 0.46
SIGMAR1 Q99720 2/20 0.46
HTR1A P08908 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
KDM4E B2RXH2 1/20 0.46
PKM P14618 1/20 0.46
CKS1B P61024 1/20 0.46
SKP1 P63208 1/20 0.46
SKP2 Q13309 1/20 0.46
CACNA1I Q9P0X4 3/20 0.45
CACNA1G O43497 1/20 0.45
CACNA1H O95180 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30840002 0.89 KCNH2 (0.51) DRD2HTR2AHTR2CKCNH2HTR2B
SCHEMBL30840016 0.82 HTR2A (0.51) DRD2HTR2AHTR2CKCNH2CACNA1I
SCHEMBL8222029 0.81 CKS1B (0.53) DRD2KDM4EPKMCKS1BSKP1
SCHEMBL29208006 0.81 HTR2A (0.54) DRD2HTR2AHTR2CKCNH2HTR2B
Hydrochloric Acid SCHEMBL29207967 0.80 HTR2A (0.53) DRD2HTR2AHTR2CKCNH2HTR2B
SCHEMBL30831997 0.79 HTR2A (0.48) DRD2HTR2AHTR2CKCNH2HTR2B
SCHEMBL30839998 0.79 HTR2A (0.46) DRD2HTR2AHTR2CKCNH2HTR2B
Hydrochloric Acid SCHEMBL29208110 0.79 HTR2A (0.52) DRD2HTR2AHTR2CKCNH2HTR2B
SCHEMBL7137625 0.79 ALDH1A1 (0.57) DRD2HTR2AHTR2CPKM
SCHEMBL29280915 0.78 HTR2A (0.61) HTR2AHTR2CKCNH2SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067302-A1 AMIDE COMPOUND AND USE THEREOF IN PREPARATION OF INHIBITOR OF SIGMA2 AND 5HT2A 瀚远医药有限公司 2024-04-04 WO disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed