SCHEMBL30831997

SCHEMBL30831997

COCC1CCC(CNC(=O)NCC2CCN(CC(=O)c3ccc(F)cc3)CC2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.48
HTR2C P28335 3/20 0.48
DRD2 P14416 2/20 0.48
HTR2B P41595 2/20 0.48
SIGMAR1 Q99720 2/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
KCNH2 Q12809 3/20 0.46
HTR1A P08908 2/20 0.45
TMEM97 Q5BJF2 1/20 0.45
ALDH1A1 P00352 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
TSHR P16473 2/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
ALOX15 P16050 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29207976 0.94 HTR2A (0.44) HTR2AHTR2CDRD2HTR2BSIGMAR1
SCHEMBL30832005 0.85 KMT2A (0.48) HTR2AHTR2CMEN1KMT2AKCNH2
Trifluoroacetic Acid SCHEMBL29208053 0.83 PTGIR (0.41) HTR2AHTR2CDRD2HTR2BSIGMAR1
Trifluoroacetic Acid SCHEMBL29207934 0.80 KMT2A (0.45) HTR2AHTR2CMEN1KMT2AKCNH2
SCHEMBL29208006 0.80 HTR2A (0.54) HTR2AHTR2CDRD2HTR2BSIGMAR1
SCHEMBL30832013 0.79 DRD2 (0.49) HTR2AHTR2CDRD2HTR2BSIGMAR1
Hydrochloric Acid SCHEMBL29207967 0.79 HTR2A (0.53) HTR2AHTR2CDRD2HTR2BSIGMAR1
Hydrochloric Acid SCHEMBL29208110 0.78 HTR2A (0.52) HTR2AHTR2CDRD2HTR2BSIGMAR1
SCHEMBL29280915 0.77 HTR2A (0.61) HTR2AHTR2CSIGMAR1KCNH2HTR1A
SCHEMBL10587379 0.77 ALDH1A1 (0.57) HTR2AHTR2CDRD2HTR2BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed