SCHEMBL30833207

SCHEMBL30833207

NC1C[C@H]2CC[C@@H](C1)N2Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.48
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
OPRM1 P35372 2/20 0.42
OPRD1 P41143 2/20 0.42
CYP3A4 P08684 2/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40
BACE1 P56817 2/20 0.40
UBE2M P61081 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
IDO1 P14902 1/20 0.39
PDE8B O95263 1/20 0.38
HSD11B1 P28845 1/20 0.38
TEAD1 P28347 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL30201771 0.91 LTA4H (0.53) LTA4HOPRM1OPRD1CYP3A4MAPT
SCHEMBL9412872 0.87 KDM4E (0.42) LTA4HKDM4EALDH1A1CYP3A4MAPT
SCHEMBL9412870 0.87 KDM4E (0.42) LTA4HKDM4EALDH1A1CYP3A4MAPT
SCHEMBL3880869 0.82 DRD2 (0.51) LTA4HMAPTMEN1KMT2A
SCHEMBL3880873 0.82 DRD2 (0.51) LTA4HMAPTMEN1KMT2A
SCHEMBL30833222 0.82 DRD2 (0.51) LTA4HMAPTMEN1KMT2A
SCHEMBL4145169 0.81 LTA4H (0.46) LTA4HKDM4EALDH1A1CYP3A4MAPT
SCHEMBL6256020 0.81 LTA4H (0.48) LTA4HKDM4EALDH1A1OPRM1OPRD1
SCHEMBL3881484 0.80 DRD2 (0.48) LTA4HKDM4EALDH1A1MAPTMAPK1
SCHEMBL3881487 0.80 DRD2 (0.48) LTA4HKDM4EALDH1A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117729914-A Serotonin 5-HT2B inhibiting compounds 硕腾服务有限责任公司 2024-03-19 CN disclosed