SCHEMBL30833265

SCHEMBL30833265

Cn1c(=O)ccc2cc(-n3ccnc3)ccc21

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.55
CYP11B2 P19099 2/20 0.55
CYP19A1 P11511 2/20 0.55
BRPF1 P55201 5/20 0.49
NCOA3 Q9Y6Q9 1/20 0.47
MAOA P21397 6/20 0.45
MAOB P27338 6/20 0.45
IDO1 P14902 1/20 0.44
CYP3A4 P08684 1/20 0.43
BAZ2B Q9UIF8 1/20 0.43
CA12 O43570 1/20 0.42
BRD4 O60885 1/20 0.42
CA9 Q16790 1/20 0.42
KAT2B Q92831 1/20 0.42
BRD9 Q9H8M2 1/20 0.42
CRBN Q96SW2 2/20 0.42
TBXAS1 P24557 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24677009 0.77 IDO1 (0.48) CYP11B1CYP11B2CYP19A1IDO1CYP3A4
SCHEMBL24677007 0.74 IDO1 (0.42) CYP11B1CYP11B2CYP19A1IDO1CYP3A4
SCHEMBL28274864 0.73 CYP11B1 (0.71) CYP11B1CYP11B2CYP19A1NCOA3MAOA
SCHEMBL7592308 0.73 CYP11B1 (0.57) CYP11B1CYP11B2CYP19A1NCOA3MAOA
SCHEMBL2071832 0.72 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1NCOA3MAOA
SCHEMBL4499181 0.70 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1NCOA3MAOA
SCHEMBL16126788 0.70 CYP11B1 (0.53) CYP11B1CYP11B2CYP19A1NCOA3MAOA
SCHEMBL10464389 0.70 CYP19A1 (0.56) CYP11B1CYP11B2CYP19A1NCOA3MAOA
SCHEMBL29766461 0.69 CD38 (0.38) CYP11B1CYP11B2NCOA3CYP3A4
SCHEMBL20538384 0.69 CYP3A4 (0.61) CYP11B1CYP11B2CYP19A1IDO1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117580829-A Quinoline and azaquinolines as inhibitors of CD38 勃林格英格翰国际有限公司 2024-02-20 CN claimed
CN-117580829-A Quinoline and azaquinolines as inhibitors of CD38 勃林格英格翰国际有限公司 2024-02-20 CN disclosed