SCHEMBL7592308

SCHEMBL7592308

Cn1ccc2ccc(-n3ccnc3)cc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.57
CYP11B2 P19099 2/20 0.57
CYP19A1 P11511 2/20 0.57
NCOA3 Q9Y6Q9 1/20 0.48
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
ENPP2 Q13822 1/20 0.46
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
NOTUM Q6P988 1/20 0.46
MAOA P21397 5/20 0.46
MAOB P27338 5/20 0.46
IDO1 P14902 1/20 0.45
CYP3A4 P08684 2/20 0.44
BAZ2B Q9UIF8 1/20 0.44
MEN1 O00255 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
KMT2A Q03164 1/20 0.44
TBXAS1 P24557 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28274864 0.74 CYP11B1 (0.71) CYP11B1CYP11B2CYP19A1NCOA3LMNA
SCHEMBL30833265 0.73 CYP11B1 (0.55) CYP11B1CYP11B2CYP19A1NCOA3MAOA
SCHEMBL2071832 0.73 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1NCOA3LMNA
SCHEMBL2532397 0.72 LMNA (0.78) CYP11B1CYP11B2CYP19A1LMNAMAPT
SCHEMBL7592382 0.71 NOTUM (0.46) LMNAMAPTNOTUMMEN1KMT2A
SCHEMBL4499181 0.71 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1NCOA3LMNA
SCHEMBL12117429 0.70 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1NCOA3LMNA
Hydrochloric Acid SCHEMBL28701756 0.70 LMNA (0.75) CYP11B1CYP11B2CYP19A1LMNAMAPT
SCHEMBL13045131 0.70 CYP19A1 (1.00) CYP11B1CYP11B2CYP19A1NCOA3LMNA
SCHEMBL15978818 0.70 CYP11B1 (0.65) CYP11B1CYP11B2CYP19A1NCOA3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242409-A2 SUBSTITUTED BISINDOLYLMALEIMIDES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-25 EP disclosed
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed
WO-2001046178-A2 SUBSTITUIERTE BISINDOLYMALEIMIDE F. HOFFMANN-LA ROCHE AG (CH) 2001-06-28 WO disclosed