SCHEMBL30833691

SCHEMBL30833691

Cn1ncc2ccc(Nc3ncc(Br)c(Nc4cccc(F)c4CS(N)(=O)=O)n3)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 6/20 0.44
SYK P43405 6/20 0.44
CDK2 P24941 4/20 0.42
JAK3 P52333 4/20 0.42
JAK2 O60674 3/20 0.42
CDC7 O00311 2/20 0.42
DAPK3 O43293 2/20 0.42
ROCK2 O75116 2/20 0.42
PRKD3 O94806 2/20 0.42
MAP4K4 O95819 2/20 0.42
PAK4 O96013 2/20 0.42
PRKACA P17612 2/20 0.42
CSNK1A1 P48729 2/20 0.42
CLK2 P49760 2/20 0.42
GSK3A P49840 2/20 0.42
GSK3B P49841 2/20 0.42
RPS6KA3 P51812 2/20 0.42
PRKX P51817 2/20 0.42
MAP4K2 Q12851 2/20 0.42
STK3 Q13188 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833673 0.86 SYK (0.45) ALKSYKCDK2JAK3JAK2
SCHEMBL29190625 0.84 SYK (0.47) ALKSYKCDK2JAK3JAK2
SCHEMBL30833701 0.80 ALK (0.68) ALKSYKCDK2JAK3JAK2
SCHEMBL29190525 0.80 ALK (0.68) ALKSYKCDK2JAK3JAK2
SCHEMBL30833810 0.78 ALK (0.49) ALKSYKCDK2JAK3JAK2
SCHEMBL29190704 0.78 ALK (0.49) ALKSYKCDK2JAK3JAK2
SCHEMBL29190577 0.78 ALK (0.55) ALKCDK9CDK7PTK2MET
SCHEMBL30833646 0.78 ALK (0.55) ALKCDK9CDK7PTK2MET
SCHEMBL30833747 0.77 ALK (0.49) ALKSYKCDK2JAK3JAK2
SCHEMBL29190613 0.77 ALK (0.49) ALKSYKCDK2JAK3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed