SCHEMBL30835697

SCHEMBL30835697

N#Cc1cc(Cl)nc2ncccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.41
ELANE P08246 5/20 0.39
CYP11B2 P19099 1/20 0.39
CLK1 P49759 1/20 0.39
CLK2 P49760 1/20 0.39
CLK3 P49761 1/20 0.39
CDK5 Q00535 1/20 0.39
DYRK1A Q13627 1/20 0.39
CDK5R1 Q15078 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
ACHE P22303 2/20 0.39
SLC40A1 Q9NP59 1/20 0.38
CCR1 P32246 1/20 0.38
CCR8 P51685 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ABCG2 Q9UNQ0 2/20 0.37
GRM4 Q14833 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL247512 0.77 L3MBTL1 (0.52) LRRK2CLK2CDK5DYRK1ACLK4
SCHEMBL1995026 0.74 LRRK2 (0.50) LRRK2ELANECLK1CLK2CLK3
SCHEMBL1577423 0.74 CCR1 (0.49) LRRK2CLK2CDK5DYRK1ACLK4
SCHEMBL12426313 0.74 KDM4E (0.44) LRRK2CLK2CDK5DYRK1ACLK4
SCHEMBL31444788 0.74 MEN1 (0.43) LRRK2CLK2CDK5DYRK1ACLK4
SCHEMBL2185260 0.74 ALDH1A1 (0.50) NCOA3DYRK1AL3MBTL1ALDH1A1
SCHEMBL27631463 0.73 CCR1 (0.45) LRRK2CYP11B2ACHECCR1CCR8
Hydrochloric Acid SCHEMBL31354904 0.73 LRRK2 (0.49) LRRK2ELANECLK1CLK2CLK3
SCHEMBL2325505 0.72 CYP11B2 (0.42) LRRK2CYP11B2CLK1CLK2CLK3
SCHEMBL25156021 0.71 NR4A2 (0.57) LRRK2NCOA3ELANECYP11B2CLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024059212-A2 6,6 WESTERN CORE COMPOUNDS AS MGLU5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME VANDERBILT UNIVERSITY (US) 2024-03-21 WO disclosed