SCHEMBL30847

SCHEMBL30847

COc1ccc2nc(NC(=O)c3cccc(OC)c3F)sc2c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 12/20 0.75
NPC1 O15118 12/20 0.75
KMT2A Q03164 8/20 0.70
MEN1 O00255 7/20 0.70
SCD O00767 5/20 0.68
POLB P06746 1/20 0.66
KLF5 Q13887 1/20 0.64
DCLK1 O15075 1/20 0.63
FES P07332 1/20 0.63
PIM1 P11309 1/20 0.63
CDK2 P24941 1/20 0.63
GSK3A P49840 1/20 0.63
GSK3B P49841 1/20 0.63
IRAK1 P51617 1/20 0.63
MAP4K2 Q12851 1/20 0.63
NTRK3 Q16288 1/20 0.63
HIPK4 Q8NE63 1/20 0.63
AURKB Q96GD4 1/20 0.63
CLK4 Q9HAZ1 1/20 0.63
STK17A Q9UEE5 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4920242 0.89 RAB9A (0.79) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL4919731 0.86 RAB9A (1.00) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL30517 0.85 RAB9A (0.82) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL30930 0.84 NPC1 (0.73) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL31005 0.83 RAB9A (0.83) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL2486652 0.83 RAB9A (0.75) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL31401 0.83 NPC1 (0.66) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL30919 0.83 RAB9A (0.72) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL4918858 0.83 RAB9A (0.76) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL16562091 0.81 RAB9A (0.78) RAB9ANPC1KMT2AMEN1SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed