SCHEMBL30853371

SCHEMBL30853371

COc1c(N2CCOCC2)ncc2[nH]ncc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.43
PIK3CD O00329 2/20 0.43
PIK3CB P42338 2/20 0.43
PDE10A Q9Y233 2/20 0.41
PIK3CG P48736 1/20 0.41
FYN P06241 1/20 0.40
PDE5A O76074 1/20 0.39
PDE6A P16499 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE3A Q14432 1/20 0.39
TRPM8 Q7Z2W7 2/20 0.39
MTOR P42345 2/20 0.39
KMT2A Q03164 2/20 0.38
MAP2K7 O14733 1/20 0.37
MEN1 O00255 1/20 0.37
PIM1 P11309 1/20 0.37
PIM3 Q86V86 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27186371 0.75 SMN1; SMN2 (0.43) PIK3CAPIK3CDPIK3CBPDE10APIK3CG
SCHEMBL27186190 0.71 ALDH1A1 (0.41) PIK3CAPIK3CDPIK3CBMTORKMT2A
SCHEMBL29844203 0.71 ALDH1A1 (0.41) PIK3CAPIK3CDPIK3CBMTORKMT2A
SCHEMBL21500052 0.69 LRRK2 (0.49) PIK3CAPDE10AFYNPDE5APDE6A
SCHEMBL19950255 0.68 BRD4 (0.40)
SCHEMBL30070507 0.68 BRD4 (0.40)
SCHEMBL4996432 0.67 LMNA (0.68) PIK3CAPIK3CDPIK3CBKMT2AMEN1
SCHEMBL26769922 0.67 KDM4E (0.64) PIK3CAPIK3CDPIK3CBPDE10AKMT2A
SCHEMBL29168322 0.66 TRPM8 (0.42) PIK3CAPIK3CDPIK3CBPDE10ATRPM8
SCHEMBL11218577 0.66 CYP2C19 (0.47) PDE10ATRPM8MTORKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117651701-A Novel substituted bicyclic aza heterocycles as SOS1 inhibitors 唯久生物技术(苏州)有限公司 2024-03-05 CN disclosed