SCHEMBL30858656

SCHEMBL30858656

Cc1c[nH]c2c(C)cc(F)cc12

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.48
REN P00797 2/20 0.46
GPR84 Q9NQS5 1/20 0.41
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
ATM Q13315 1/20 0.34
TDO2 P48775 1/20 0.32
SYK P43405 3/20 0.32
TRIM24 O15164 1/20 0.32
TRIM33 Q9UPN9 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
BRPF1 P55201 1/20 0.31
MAPT P10636 1/20 0.31
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15730096 0.85 GPR84 (0.58) ARRENGPR84ALDH1A1LMNA
SCHEMBL15389028 0.82 REN (0.49) ARRENGPR84ALDH1A1LMNA
SCHEMBL1137433 0.82 REN (0.43) ARRENGPR84ALDH1A1LMNA
SCHEMBL23685894 0.79 REN (0.41) ARRENGPR84ALDH1A1LMNA
SCHEMBL16727212 0.79 REN (0.41) ARRENGPR84ALDH1A1LMNA
SCHEMBL671315 0.77 TRIM24 (0.56) ARGPR84ALDH1A1LMNATRIM24
SCHEMBL20688241 0.77 MAPT (0.50) ARRENATMTRIM24TRIM33
SCHEMBL18299455 0.75 KIF11 (0.37) ARRENATMCYP1A2MAPT
SCHEMBL16571178 0.75 REN (0.47) ARRENGPR84ATM
SCHEMBL31223258 0.75 AR (0.41) ARGPR84ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4580621-A2 T-TYPE VOLTAGE-GATED CALCIUM CHANNEL POTENTIATORS The Broad Institute, Inc. (US) 2025-07-09 EP disclosed
CN-120091815-A T-type voltage-gated calcium channel enhancer 广泛研究所股份有限公司 2025-06-03 CN disclosed
WO-2024050312-A2 T-TYPE VOLTAGE-GATED CALCIUM CHANNEL POTENTIATORS THE BROAD INSTITUTE, INC. (US) 2024-03-07 WO disclosed