SCHEMBL30876355

SCHEMBL30876355

c1ccc2c(c1)nc1n(-c3ccc4[nH]c5ccccc5c4c3)c3ccccc3n21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.40
AHR P35869 1/20 0.39
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 3/20 0.36
GPR3 P46089 1/20 0.36
KDM4E B2RXH2 5/20 0.35
KIF11 P52732 3/20 0.35
HPGD P15428 3/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GABRP O00591 3/20 0.35
GABRD O14764 3/20 0.35
GABRA1 P14867 3/20 0.35
GABRB1 P18505 3/20 0.35
GABRG2 P18507 3/20 0.35
GABRB3 P28472 3/20 0.35
GABRA5 P31644 3/20 0.35
GABRA3 P34903 3/20 0.35
GABRA2 P47869 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12800982 1.00 TOP2A (0.40) TOP2AAHRALDH1A1HSD17B10GPR3
SCHEMBL15631669 0.94 KDM4E (0.35) TOP2AAHRALDH1A1HSD17B10KDM4E
SCHEMBL23219318 0.92 TOP2A (0.40) TOP2AAHRALDH1A1HSD17B10GPR3
SCHEMBL26342598 0.85 CDK4 (0.36) TOP2AALDH1A1HSD17B10KDM4EHPGD
SCHEMBL18830921 0.83 TOP2A (0.36) TOP2AAHRALDH1A1HSD17B10GPR3
SCHEMBL18687112 0.83 HPGD (0.37) TOP2AAHRALDH1A1HSD17B10KDM4E
SCHEMBL18698129 0.83 HPGD (0.37) TOP2AAHRALDH1A1HSD17B10KDM4E
SCHEMBL20616762 0.82 TOP2A (0.41) TOP2AAHRALDH1A1HSD17B10GPR3
SCHEMBL18934348 0.82 TOP2A (0.41) TOP2AAHRALDH1A1HSD17B10GPR3
SCHEMBL23652412 0.82 ADORA2B (0.35) TOP2AAHRALDH1A1HSD17B10GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024033282-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2024-02-15 WO disclosed