SCHEMBL30877293

SCHEMBL30877293

COC(=O)c1cc2cc(C#N)cnc2n1S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD1 Q9Y239 4/20 0.43
NOD2 Q9HC29 3/20 0.43
CCR6 P51684 3/20 0.42
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35
POLB P06746 1/20 0.35
ENPP3 O14638 1/20 0.35
ENPP1 P22413 1/20 0.35
ALOX5 P09917 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23147752 0.85 NOD2 (0.47) NOD1NOD2CCR6KDM4ELMNA
SCHEMBL23148046 0.81 NOD1 (0.48) NOD1NOD2KDM4ELMNATSHR
SCHEMBL23147626 0.78 CYP11B1 (0.44) NOD1NOD2CYP11B1CYP11B2OPRM1
SCHEMBL29813550 0.77 NOD1 (0.45) NOD1NOD2L3MBTL1OPRM1OPRD1
SCHEMBL23147751 0.77 NOD1 (0.45) NOD1NOD2L3MBTL1OPRM1OPRD1
SCHEMBL30877335 0.76 KDM4E (0.40) NOD1NOD2CCR6KDM4ELMNA
SCHEMBL30877374 0.76 CCR6 (0.37) CCR6KDM4ELMNATSHRL3MBTL1
SCHEMBL23147551 0.75 NOD1 (0.47) NOD1NOD2KDM4ELMNATSHR
SCHEMBL9378689 0.74 NOD2 (0.55) NOD1NOD2KDM4ELMNATSHR
SCHEMBL2927020 0.74 PTGS2 (0.42) NOD1NOD2KDM4ELMNAPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964643-B Pyrrole [2,3-b ] pyridine derivative and preparation method and application thereof 苏州朗睿生物医药有限公司 2024-07-02 CN disclosed
CN-117964643-A Pyrrole [2,3-b ] pyridine derivative and preparation method and application thereof 苏州朗睿生物医药有限公司 2024-05-03 CN disclosed