SCHEMBL30883146

SCHEMBL30883146

Cc1ccc(Cl)cc1N1CCN(c2ccc(C(=O)O)cc2NC(=O)c2ccc(Cl)cc2)CC1

nearest known ligand 0.88

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 4/20 0.88
MEN1 O00255 4/20 0.55
KMT2A Q03164 4/20 0.55
IDH2 P48735 1/20 0.54
LMNA P02545 1/20 0.53
MAPT P10636 3/20 0.52
TP53 P04637 2/20 0.52
POLB P06746 2/20 0.52
ALDH1A1 P00352 3/20 0.52
NPSR1 Q6W5P4 1/20 0.52
HTT P42858 1/20 0.52
MCL1 Q07820 1/20 0.52
KDM4E B2RXH2 2/20 0.51
ALOX15 P16050 1/20 0.51
MAPK1 P28482 1/20 0.51
TDP1 Q9NUW8 1/20 0.50
USP2 O75604 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29204805 1.00 XPO1 (0.88) XPO1MEN1KMT2AIDH2LMNA
SCHEMBL29204831 0.94 XPO1 (0.77) XPO1MEN1KMT2AIDH2LMNA
SCHEMBL30883139 0.94 XPO1 (0.77) XPO1MEN1KMT2AIDH2LMNA
SCHEMBL30883142 0.93 XPO1 (1.00) XPO1MEN1KMT2AIDH2LMNA
SCHEMBL29204833 0.93 XPO1 (1.00) XPO1MEN1KMT2AIDH2LMNA
SCHEMBL29204835 0.92 XPO1 (0.74) XPO1MEN1KMT2AIDH2LMNA
SCHEMBL29204842 0.90 XPO1 (0.80) XPO1MEN1KMT2AMAPTTP53
SCHEMBL29204810 0.89 XPO1 (0.70) XPO1KMT2AIDH2LMNAMAPT
SCHEMBL30883143 0.88 XPO1 (0.69) XPO1MEN1KMT2ALMNAMAPT
SCHEMBL29204830 0.88 XPO1 (0.69) XPO1MEN1KMT2ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964578-A Non-covalent CRM1 inhibitor and preparation method and application thereof 四川大学 2024-05-03 CN disclosed