SCHEMBL29204830

SCHEMBL29204830

O=C(O)c1ccc(N2CCN(c3cc(Cl)ccc3Cl)CC2)c(NC(=O)c2ccc(Cl)cc2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 4/20 0.69
KMT2A Q03164 5/20 0.58
MEN1 O00255 4/20 0.58
ALDH1A1 P00352 4/20 0.54
NPSR1 Q6W5P4 3/20 0.54
HTT P42858 2/20 0.53
MCL1 Q07820 1/20 0.53
MAPT P10636 4/20 0.53
LMNA P02545 2/20 0.53
MAPK1 P28482 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
APOBEC3G Q9HC16 1/20 0.51
KDM4E B2RXH2 2/20 0.50
HPGD P15428 2/20 0.50
ALOX15 P16050 1/20 0.50
TP53 P04637 2/20 0.49
POLB P06746 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
SERPINE1 P05121 1/20 0.49
HDAC1 Q13547 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30883143 1.00 XPO1 (0.69) XPO1KMT2AMEN1ALDH1A1NPSR1
SCHEMBL30883146 0.88 XPO1 (0.88) XPO1KMT2AMEN1ALDH1A1NPSR1
SCHEMBL29204805 0.88 XPO1 (0.88) XPO1KMT2AMEN1ALDH1A1NPSR1
SCHEMBL29204806 0.87 WDR5 (0.61) XPO1KMT2AMEN1ALDH1A1HTT
SCHEMBL30883141 0.85 XPO1 (0.66) XPO1KMT2AMEN1NPSR1HTT
SCHEMBL29204829 0.85 XPO1 (0.66) XPO1KMT2AMEN1NPSR1HTT
SCHEMBL29204831 0.82 XPO1 (0.77) XPO1KMT2AMEN1ALDH1A1NPSR1
SCHEMBL30883139 0.82 XPO1 (0.77) XPO1KMT2AMEN1ALDH1A1NPSR1
SCHEMBL30883142 0.82 XPO1 (1.00) XPO1KMT2AMEN1ALDH1A1NPSR1
SCHEMBL29204833 0.82 XPO1 (1.00) XPO1KMT2AMEN1ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964578-A Non-covalent CRM1 inhibitor and preparation method and application thereof 四川大学 2024-05-03 CN disclosed