SCHEMBL3089392

SCHEMBL3089392

c1ccc(N=Nc2cccc3cc4ccccc4cc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 8/20 0.46
KMT2A Q03164 8/20 0.46
MAPK1 P28482 4/20 0.46
TDP1 Q9NUW8 4/20 0.46
NPC1 O15118 4/20 0.46
MAPT P10636 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
CYP3A4 P08684 3/20 0.41
HBB P68871 2/20 0.41
TSHR P16473 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CHRM1 P11229 1/20 0.41
CYP2C9 P11712 1/20 0.41
DRD2 P14416 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30139030 0.90 SIGMAR1 (0.45) ALDH1A1MEN1KMT2AMAPK1TDP1
SCHEMBL28961947 0.86 SENP7 (0.47) ALDH1A1MEN1KMT2AMAPK1TDP1
SCHEMBL29978043 0.86 SENP7 (0.47) ALDH1A1MEN1KMT2AMAPK1TDP1
SCHEMBL348429 0.82 SIGMAR1 (0.41) ALDH1A1MEN1KMT2AMAPK1TDP1
SCHEMBL2926928 0.82 MEN1 (0.55) ALDH1A1MEN1KMT2AMAPK1TDP1
Azobenzene SCHEMBL11226032 0.82 MEN1 (0.55) ALDH1A1MEN1KMT2AMAPK1TDP1
SCHEMBL2926925 0.82 MEN1 (0.55) ALDH1A1MEN1KMT2AMAPK1TDP1
Azobenzene SCHEMBL11130609 0.82 MEN1 (0.55) ALDH1A1MEN1KMT2AMAPK1TDP1
SCHEMBL9017635 0.81 SENP7 (0.42) ALDH1A1MEN1KMT2AMAPK1TDP1
SCHEMBL23257776 0.80 MEN1 (0.53) ALDH1A1MEN1KMT2AMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025134143-A1 A METHOD FOR THE SYNTHESIS OF SUBSTITUTED ANTHRANILIC AMIDE COMPOUNDS, INTERMEDIATES AND SALTS THEREOF PI INDUSTRIES LTD. (IN) 2025-06-26 WO claimed
WO-2025134143-A1 A METHOD FOR THE SYNTHESIS OF SUBSTITUTED ANTHRANILIC AMIDE COMPOUNDS, INTERMEDIATES AND SALTS THEREOF PI INDUSTRIES LTD. (IN) 2025-06-26 WO disclosed
EP-4330223-A1 HYDROGENATION OF NITROBENZOIC ACID AND NITROBENZAMIDE FMC CORPORATION (US) 2024-03-06 EP disclosed
WO-2024025285-A1 CARBOXAMIDE DERIVATIVE OF TRIAZINYL FUSED RING, AND NEMATICIDAL USE THEREOF 한국화학연구원 2024-02-01 WO disclosed
EP-4308121-A1 THERAPEUTIC CONJUGATES Totus Medicines Inc. (US) 2024-01-24 EP disclosed
WO-2022232366-A1 HYDROGENATION OF NITROBENZOIC ACID AND NITROBENZAMIDE FMC CORPORATION (US) 2022-11-03 WO disclosed
WO-2022198024-A1 THERAPEUTIC CONJUGATES TOTUS MEDICINES INC. (US) 2022-09-22 WO disclosed
EP-4033900-A1 ANTHRANILAMIDE COMPOSITION FMC CORPORATION (US) 2022-08-03 EP disclosed
WO-2021097118-A1 SMALL TYPE II CAS PROTEINS AND METHODS OF USE THEREOF THE BROAD INSTITUTE, INC. (US) 2021-05-20 WO disclosed
WO-2021064731-A1 PESTICIDAL MIXTURES ADAMA MAKHTESHIM LTD. (IL) 2021-04-08 WO disclosed
WO-2009055239-A1 BORDETELLA DETECTION ASSAY QUEST DIAGNOSTICS INVESTMENTS INCORPORATED (US) 2009-04-30 WO disclosed
JP-2009013158-A PRODUCTION METHOD OF ANTHRANIL AMIDE COMPOUND ISHIHARA SANGYO KAISHA LTD 2009-01-22 JP disclosed
JP-2009013158-A PRODUCTION METHOD OF ANTHRANIL AMIDE COMPOUND ISHIHARA SANGYO KAISHA LTD 2009-01-22 JP disclosed
WO-2008082502-A2 PROCESS FOR PREPARING 2-AMINO-5-CYANOBENZOIC ACID DERIVATIVES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2008-07-10 WO disclosed
WO-2008069990-A1 LIQUID FORMULATIONS OF CARBOXAMIDE ARTHROPODICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2008-06-12 WO disclosed
WO-2007070680-A2 OPTICALLY DETECTABLE PROBES FOR IDENTIFICATION AND TREATMENT OF TUMORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2007-06-21 WO disclosed
US-20050161863-A1 Method for the direct and continuous production of hollow articles from a polymer melt ZIMMER AKTIENGESELLSCHAFT 2005-07-28 US disclosed
CN-1538836-A Substituted amine derivatives and method of use ������������� 2004-10-20 CN disclosed
EP-0320281-A2 Corrosion inhibitor EXXON RESEARCH AND ENGINEERING COMPANY (US) 1989-06-14 EP disclosed
US-3818001-A 1,2,3-BENZOTRIAZIN-4(3H)-ONES SANDOZ AG 1974-06-18 US disclosed