SCHEMBL30895265

SCHEMBL30895265

Cc1nn(C(F)(F)F)c2cc(O)ccc12

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.40
CYP19A1 P11511 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
KMO O15229 1/20 0.35
HSD17B3 P37058 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
KCNJ11 Q14654 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
RIPK2 O43353 1/20 0.32
KDR P35968 1/20 0.32
MAPK14 Q16539 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30895272 0.80 PDGFRA (0.38) CYP19A1CYP2C9CYP11B1CYP11B2KMO
SCHEMBL30895271 0.80 PDGFRA (0.38) CYP19A1CYP2C9CYP11B1CYP11B2KMO
SCHEMBL15730578 0.75 ESR1 (0.60) ESR1KMOADORA2AADORA2B
SCHEMBL30895262 0.72 KDM4E (0.31)
SCHEMBL15723742 0.71 GRM4 (0.43) ESR1KDRHTT
SCHEMBL18853871 0.71 ESR1 (0.63) ESR1KMOSLC22A12ADORA2AADORA2B
SCHEMBL30895264 0.71 IRAK4 (0.40)
SCHEMBL176951 0.70 ELANE (0.42) ESR1KMOSLC22A12HTT
SCHEMBL30895267 0.70 MAPK8 (0.39) CYP2C9ADORA2AADORA2BHTT
SCHEMBL176840 0.67 ESR2 (0.41) ESR1KMOSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4608507-A1 COMPOUNDS AND COMPOSITIONS AS GPR52 MODULATORS Neurocrine Biosciences, Inc. (US) 2025-09-03 EP disclosed
WO-2024091538-A1 COMPOUNDS AND COMPOSITIONS AS GPR52 MODULATORS NEUROCRINE BIOSCIENCES, INC. (US) 2024-05-02 WO disclosed