SCHEMBL3089669

SCHEMBL3089669

C=CC(NCCc1c[nH]c2ccccc12)P(=O)(O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
PKM P14618 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
BLM P54132 1/20 0.51
SIRT1 Q96EB6 4/20 0.50
HTR2A P28223 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HTR1A P08908 1/20 0.50
HTT P42858 1/20 0.50
MMP9 P14780 1/20 0.49
AANAT Q16613 1/20 0.49
MC5R P33032 1/20 0.49
MC3R P41968 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3080644 0.85 HTR2C (0.55) MEN1KMT2ALMNACYP1A2TSHR
SCHEMBL3082092 0.77 ALOX15 (0.57) MMP9
SCHEMBL3082097 0.77 ALOX15 (0.57) MMP9
SCHEMBL2989714 0.77 MC5R (0.64) MEN1KMT2ANPC1RAB9ALMNA
Phosphoric Acid SCHEMBL28038796 0.76 MEN1 (0.62) MEN1KMT2ANPC1RAB9ALMNA
SCHEMBL3192955 0.76 HTR1A (0.54) LMNAHTR2AALDH1A1HTR1AHTT
SCHEMBL21781048 0.73 KDM4E (0.65) MEN1KMT2ANPC1RAB9ALMNA
SCHEMBL2732463 0.73 HTR2A (0.69) MEN1KMT2ALMNACYP1A2PKM
SCHEMBL30536673 0.73 HTR2A (0.69) MEN1KMT2ALMNACYP1A2PKM
SCHEMBL21943192 0.73 HTR2A (0.64) MEN1KMT2ANPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100247463-A1 N-(PHOSPHONOALKYL)-AMINO ACIDS, DERIVATIVES THEREOF AND COMPOSITIONS AND METHODS OF USE YU RUEY J 2010-09-30 US disclosed
US-7776844-B2 N-(phosphonoalkyl)-amino acids, derivatives thereof and compositions and methods of use YU RUEY J 2010-08-17 US disclosed
US-20090208499-A1 N-(Phosphonoalkyl)-Amino Acids, Derivatives Thereof and Compositions and Methods of Use YU RUEY J 2009-08-20 US disclosed
US-7572776-B2 N-(phosphonoalkyl)-amino acids, derivatives thereof and compositions and methods of use YU RUEY J 2009-08-11 US disclosed
US-20080306025-A1 N-(PHOSPHONOALKYL)-AMINO ACIDS, DERIVATIVES THEREOF AND COMPOSITIONS AND METHODS OF USE YU RUEY J 2008-12-11 US disclosed
US-7429575-B2 N-(phosphonoalkyl)-amino acids, derivatives thereof and compositions and methods of use YU RUEY J 2008-09-30 US disclosed
US-20070161543-A1 N-(PHOSPHONOALKYL)-AMINO ACIDS, DERIVATIVES THEREOF AND COMPOSITIONS AND METHODS OF USE YU RUEY J 2007-07-12 US disclosed