SCHEMBL30901296

SCHEMBL30901296

FC(F)(F)c1c(Br)ncc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
GPR3 P46089 1/20 0.42
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
ULK1 O75385 1/20 0.34
TRPM8 Q7Z2W7 2/20 0.33
HPGD P15428 1/20 0.33
AURKA O14965 1/20 0.32
ERBB2 P04626 1/20 0.32
KDR P35968 1/20 0.32
TDP1 Q9NUW8 3/20 0.32
CNR2 P34972 2/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
GLA P06280 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21954998 1.00 KDM4E (0.42) KDM4EGPR3MAPTL3MBTL1CYP11B1
SCHEMBL15611267 0.78 KDM4E (0.42) KDM4EGPR3MAPTCYP11B1CYP11B2
SCHEMBL12526215 0.78 GPR3 (0.42) KDM4EGPR3MAPTL3MBTL1CYP11B1
SCHEMBL4105404 0.78 KDM4E (0.42) KDM4EGPR3MAPTCYP11B1CYP11B2
SCHEMBL30901299 0.78 KDM4E (0.42) KDM4EGPR3MAPTCYP11B1CYP11B2
SCHEMBL22037342 0.75 KDM4E (0.40) KDM4EGPR3MAPTL3MBTL1CYP11B1
SCHEMBL16552260 0.74 KDM4E (0.50) KDM4EGPR3MAPTL3MBTL1TDP1
SCHEMBL30901311 0.74 KDM4E (0.50) KDM4EGPR3MAPTL3MBTL1TDP1
SCHEMBL24390567 0.74 KDM4E (0.39) KDM4EGPR3MAPTL3MBTL1CYP11B1
SCHEMBL22016872 0.74 KDM4E (0.39) KDM4EGPR3CYP11B1CYP11B2ULK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119462635-A Quinoline derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2025-02-18 CN disclosed
CN-112969687-B Quinoline derivatives as a4 b 7 integrin inhibitors 吉利德科学公司 2024-08-23 CN disclosed
CN-112969700-B Imidazopyridine derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2024-08-20 CN disclosed
CN-112996786-B Compounds for inhibiting alpha 4 beta 7 integrin 吉利德科学公司 2024-08-20 CN disclosed
CN-112969504-B Compounds for inhibiting alpha 4 beta 7 integrin 吉利德科学公司 2024-04-09 CN disclosed