SCHEMBL30901299

SCHEMBL30901299

Nc1ncc2ccccc2c1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
GPR3 P46089 1/20 0.42
BACE1 P56817 2/20 0.41
F12 P00748 1/20 0.41
PLAU P00749 1/20 0.41
NCF1 P14598 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
PDPK1 O15530 1/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TSHR P16473 1/20 0.38
KEAP1 Q14145 1/20 0.38
USP7 Q93009 1/20 0.37
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15611267 1.00 KDM4E (0.42) KDM4EGPR3BACE1F12PLAU
SCHEMBL20989876 0.81 KDM4E (0.42) KDM4EGPR3BACE1F12PLAU
SCHEMBL12490356 0.80 KDM4E (0.41) KDM4EGPR3BACE1F12PLAU
SCHEMBL12490232 0.79 KDM4E (0.40) KDM4EGPR3BACE1F12PLAU
SCHEMBL21954998 0.78 KDM4E (0.42) KDM4EGPR3BACE1ALDH1A1HPGD
SCHEMBL12526215 0.78 GPR3 (0.42) KDM4EGPR3BACE1ALDH1A1HPGD
SCHEMBL4105404 0.78 KDM4E (0.42) KDM4EGPR3ALDH1A1CYP3A4HPGD
SCHEMBL30901296 0.78 KDM4E (0.42) KDM4EGPR3BACE1ALDH1A1HPGD
SCHEMBL22037342 0.75 KDM4E (0.40) KDM4EGPR3CYP3A4HPGDTSHR
SCHEMBL28301397 0.74 KDM4E (0.50) KDM4EGPR3BACE1F12PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119462635-A Quinoline derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2025-02-18 CN disclosed
CN-112969687-B Quinoline derivatives as a4 b 7 integrin inhibitors 吉利德科学公司 2024-08-23 CN disclosed
CN-112969700-B Imidazopyridine derivatives as alpha 4 beta 7 integrin inhibitors 吉利德科学公司 2024-08-20 CN disclosed
CN-112996786-B Compounds for inhibiting alpha 4 beta 7 integrin 吉利德科学公司 2024-08-20 CN disclosed
CN-112969504-B Compounds for inhibiting alpha 4 beta 7 integrin 吉利德科学公司 2024-04-09 CN disclosed