SCHEMBL30912436

SCHEMBL30912436

O=c1c(Br)cccn1C1CCOCC1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.38
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM1 P11229 1/20 0.36
CYP2A13 Q16696 1/20 0.36
DHODH Q02127 3/20 0.35
HSD17B3 P37058 1/20 0.35
TYK2 P29597 9/20 0.33
PIK3CA P42336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30912557 0.88 DHODH (0.40) DHODHTYK2
SCHEMBL19531954 0.84 IL4I1 (0.39) HCAR1DHODH
SCHEMBL28462395 0.83 TYK2 (0.33) CYP2A13DHODHTYK2
SCHEMBL22051977 0.81 TYK2 (0.38) TYK2
SCHEMBL20688017 0.80 HCAR1 (0.38) HCAR1CHRM2CHRM4CHRM1DHODH
SCHEMBL21659036 0.78 HCAR1 (0.40) HCAR1CHRM2CHRM4CHRM1DHODH
SCHEMBL21659038 0.76 TYK2 (0.36) HCAR1CHRM2CHRM4CHRM1DHODH
SCHEMBL20687697 0.76 TYK2 (0.46) TYK2
SCHEMBL21246029 0.76 CNR2 (0.39) TYK2
SCHEMBL17682621 0.74 P2RX7 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4619406-A1 TRICYCLIC COMPOUNDS Schrödinger, Inc. (US) 2025-09-24 EP disclosed
CN-118843626-A Heterocyclic compounds as DYRK1A inhibitors 普罗塞纳生物科学有限公司 2024-10-25 CN disclosed
WO-2024107393-A1 TRICYCLIC COMPOUNDS SCHRÖDINGER, INC. (US) 2024-05-23 WO disclosed