SCHEMBL30916147

SCHEMBL30916147

CC(=O)N1CCc2c(nc(C(N)=O)n2C)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 4/20 0.39
BRD4 O60885 2/20 0.39
GRM5 P41594 1/20 0.39
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
BAZ2B Q9UIF8 2/20 0.38
BPTF Q12830 1/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
NOTUM Q6P988 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
BTK Q06187 1/20 0.35
DPP4 P27487 2/20 0.34
DPP8 Q6V1X1 2/20 0.34
DPP7 Q9UHL4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28579456 0.87 GRM5 (0.40) CREBBPBRD4GRM5BAZ2BPIK3R1
SCHEMBL23611067 0.83 PDCD1 (0.46) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL23374970 0.80 CCR5 (0.42) CREBBPBRD4GRM5BAZ2BPIK3R1
SCHEMBL29716001 0.78 PDCD1 (0.41) ALDH1A1L3MBTL1PIK3R1PIK3CAMEN1
SCHEMBL30340518 0.78 PDCD1 (0.43) ALDH1A1L3MBTL1MEN1KMT2AKDM4E
SCHEMBL30703775 0.77 PDCD1 (0.42) PDCD1CD274DPP4CNR2
SCHEMBL29933269 0.77 CNR2 (0.43) PIK3R1PIK3CAPDCD1CD274DPP4
SCHEMBL29022800 0.77 PDCD1 (0.52) PDCD1CD274
SCHEMBL28508015 0.77 DPP4 (0.35) DPP4
SCHEMBL30966759 0.76 PDCD1 (0.39) PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111936475-B Immunomodulator, composition and preparation method thereof 贝达药业股份有限公司 2024-05-10 CN claimed
CN-111936475-B Immunomodulator, composition and preparation method thereof 贝达药业股份有限公司 2024-05-10 CN disclosed