SCHEMBL30935565

SCHEMBL30935565

Cc1ccc(Cc2nc(-c3ccc(C)c(N)c3)no2)cc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.66
SMN1; SMN2 Q16637 7/20 0.66
TDP1 Q9NUW8 7/20 0.66
NPC1 O15118 6/20 0.66
MAPK1 P28482 5/20 0.66
TSHR P16473 4/20 0.66
L3MBTL1 Q9Y468 6/20 0.56
KMT2A Q03164 4/20 0.55
MEN1 O00255 3/20 0.55
S1PR1 P21453 1/20 0.55
ALDH1A1 P00352 2/20 0.54
LMNA P02545 3/20 0.51
HTT P42858 2/20 0.49
ALOX15 P16050 1/20 0.47
ATM Q13315 1/20 0.46
MAPT P10636 1/20 0.46
KDM4E B2RXH2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31261554 0.90 RAB9A (0.66) RAB9ASMN1; SMN2TDP1NPC1MAPK1
SCHEMBL31261572 0.77 LMNA (0.52) RAB9ASMN1; SMN2TDP1NPC1MAPK1
SCHEMBL30935486 0.76 SCN5A (0.44) RAB9ASMN1; SMN2TDP1NPC1MAPK1
SCHEMBL14327884 0.76 S1PR1 (0.70) RAB9ASMN1; SMN2TDP1NPC1MAPK1
SCHEMBL26005529 0.76 L3MBTL1 (0.70) RAB9ASMN1; SMN2TDP1NPC1MAPK1
SCHEMBL31013417 0.75 L3MBTL1 (0.61) RAB9ANPC1TSHRL3MBTL1S1PR1
SCHEMBL3250198 0.75 L3MBTL1 (0.61) RAB9ANPC1TSHRL3MBTL1S1PR1
SCHEMBL19131277 0.75 NPC1 (0.60) RAB9ASMN1; SMN2TDP1NPC1MAPK1
SCHEMBL14741559 0.74 TP53 (0.50) RAB9ASMN1; SMN2NPC1MAPK1TSHR
SCHEMBL14741772 0.74 TP53 (0.44) RAB9ASMN1; SMN2TDP1NPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4630424-A1 COMPOUNDS AND COMPOSITIONS AS C-KIT KINASE INHIBITORS Third Harmonic Bio, Inc. (US) 2025-10-15 EP disclosed
US-20240254119-A1 COMPOUNDS AND COMPOSITIONS AS c-Kit KINASE INHIBITORS Calixis Inc. 2024-08-01 US disclosed
WO-2024124002-A1 COMPOUNDS AND COMPOSITIONS AS C-KIT KINASE INHIBITORS THIRD HARMONIC BIO, INC. (US) 2024-06-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240254119-A1 COMPOUNDS AND COMPOSITIONS AS c-Kit KINASE INHIBITORS KIT, AURKC, PRKCE RAB9A 1260/4885SMN1; SMN2 4236/4885TDP1 3217/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.