SCHEMBL30935664

SCHEMBL30935664

CCOC(=O)c1cnc2cc(-c3cscn3)ccn12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
GLA P06280 2/20 0.46
HPGD P15428 1/20 0.46
IDO1 P14902 5/20 0.43
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.40
TGFBR1 P36897 2/20 0.40
CDC7 O00311 1/20 0.39
DBF4 Q9UBU7 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30935669 0.84 TGFBR1 (0.51) GAAKDM4EGLAIDO1RAB9A
SCHEMBL30935504 0.83 JMJD6 (0.51) GAAALDH1A1KDM4EGLAHPGD
SCHEMBL14738480 0.82 KDM4E (0.49) GAAALDH1A1KDM4EGLAHPGD
SCHEMBL30935693 0.82 KDM4A (0.43) GAAALDH1A1KDM4ERAB9ANPC1
SCHEMBL17437898 0.81 KDR (0.51) GAAALDH1A1KDM4EGLAHPGD
SCHEMBL2051512 0.79 GAA (0.53) GAAALDH1A1KDM4EGLAHPGD
SCHEMBL14742881 0.79 KDM4E (0.70) GAAALDH1A1KDM4EGLAHPGD
SCHEMBL9941870 0.78 KDM4E (0.54) GAAALDH1A1KDM4EGLAHPGD
SCHEMBL19128510 0.77 FLT3 (0.53) GAAALDH1A1KDM4EGLAHPGD
SCHEMBL16370033 0.77 KDM4E (0.53) GAAALDH1A1KDM4EGLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4630423-A1 COMPOUNDS AND COMPOSITIONS AS C-KIT KINASE INHIBITORS Third Harmonic Bio, Inc. (US) 2025-10-15 EP disclosed
EP-4630424-A1 COMPOUNDS AND COMPOSITIONS AS C-KIT KINASE INHIBITORS Third Harmonic Bio, Inc. (US) 2025-10-15 EP disclosed
WO-2024123966-A1 COMPOUNDS AND COMPOSITIONS AS C-KIT KINASE INHIBITORS THIRD HARMONIC BIO, INC. (US) 2024-06-13 WO disclosed
WO-2024124002-A1 COMPOUNDS AND COMPOSITIONS AS C-KIT KINASE INHIBITORS THIRD HARMONIC BIO, INC. (US) 2024-06-13 WO disclosed