SCHEMBL30944307

SCHEMBL30944307

CC12CC3CC(C)(C1)CC(C(=O)Nc1nc4ccc(Cl)cc4o1)(C3)C2

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.44
ALOX15 P16050 1/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
NPC1 O15118 1/20 0.42
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
S1PR3 Q99500 1/20 0.40
FBP1 P09467 2/20 0.39
EPHX2 P34913 1/20 0.39
CSNK1D P48730 2/20 0.39
FFAR2 O15552 1/20 0.39
CSNK1E P49674 1/20 0.38
BACE1 P56817 1/20 0.37
ANO1 Q5XXA6 1/20 0.37
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30944413 0.92 FFAR2 (0.47) P2RX7ALOX15GAAHTTNPC1
SCHEMBL30944418 0.88 GAA (0.43) P2RX7ALOX15GAAHTTNPC1
SCHEMBL31236385 0.87 P2RX7 (0.48) P2RX7ALOX15GAAHTTNPC1
SCHEMBL30944358 0.86 NPC1 (0.42) P2RX7ALOX15GAAHTTNPC1
SCHEMBL28525120 0.85 ALOX15 (0.41) P2RX7ALOX15GAAHTTNPC1
SCHEMBL30944317 0.85 NPC1 (0.47) P2RX7ALOX15GAAHTTNPC1
SCHEMBL30944396 0.83 ALOX15 (0.47) P2RX7ALOX15GAAHTTNPC1
SCHEMBL30944379 0.81 P2RX7 (0.47) P2RX7ALOX15GAAHTTNPC1
SCHEMBL30944383 0.77 DYRK1A (0.56) NPC1KMT2APOLBRAB9A
SCHEMBL30944369 0.76 GAA (0.44) P2RX7ALOX15GAAHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed