SCHEMBL30948604

SCHEMBL30948604

CP(C)c1ccccc1Nc1ccnc(Nc2ccc(F)c([N+](=O)[O-])c2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 12/20 0.51
AURKB Q96GD4 8/20 0.51
MAPK8 P45983 7/20 0.51
PIM1 P11309 3/20 0.51
GSK3B P49841 3/20 0.51
CLK4 Q9HAZ1 3/20 0.51
CDK2 P24941 3/20 0.51
HIPK2 Q9H2X6 2/20 0.51
MAP4K4 O95819 1/20 0.51
MKNK2 Q9HBH9 1/20 0.51
IRAK4 Q9NWZ3 1/20 0.51
DAPK3 O43293 2/20 0.48
JAK2 O60674 2/20 0.48
PRKD3 O94806 2/20 0.48
CSNK1A1 P48729 2/20 0.48
CDK8 P49336 2/20 0.48
CLK2 P49760 2/20 0.48
GSK3A P49840 2/20 0.48
CDK9 P50750 2/20 0.48
RPS6KA3 P51812 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30948603 1.00 AURKA (0.51) AURKAAURKBMAPK8PIM1GSK3B
SCHEMBL30948599 0.84 GLO1 (0.48) AURKAAURKBMAPK8GSK3BCLK4
SCHEMBL29253649 0.84 GLO1 (0.48) AURKAAURKBMAPK8GSK3BCLK4
SCHEMBL655435 0.84 NPC1 (0.55) AURKAAURKBMAPK8PIM1GSK3B
SCHEMBL22520126 0.83 AURKA (0.48) AURKAAURKBMAPK8PIM1GSK3B
SCHEMBL30948608 0.83 EGFR (0.50) AURKAAURKBMAPK8PIM1GSK3B
SCHEMBL28665507 0.82 MAPK9 (0.46) AURKAAURKBGSK3BCDK2CDK9
SCHEMBL30948627 0.77 ABCG2 (0.46) AURKAAURKBMAPK8PIM1GSK3B
SCHEMBL656702 0.73 ALDH1A1 (0.65) AURKAAURKBMAPK8PIM1GSK3B
SCHEMBL29190558 0.72 ULK1 (0.45) AURKAGSK3BCDK2JAK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677680-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2024-05-10 CN disclosed