SCHEMBL30948965

SCHEMBL30948965

Cc1nc(N[C@@H]2CN(C(=O)OCc3ccccc3)CC23CC3)ccc1-c1cn2c(n1)C(F)(F)CC2

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 6/20 0.36
KDM1A O60341 2/20 0.35
F13A1 P00488 1/20 0.34
TGM2 P21980 1/20 0.34
TGM1 P22735 1/20 0.34
CNR2 P34972 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ENPP2 Q13822 2/20 0.33
RORC P51449 2/20 0.33
TRPC3 Q13507 1/20 0.33
TRPC7 Q9HCX4 1/20 0.33
ACACB O00763 1/20 0.33
USP30 Q70CQ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31634667 1.00 GRIN2B (0.36) GRIN2BKDM1AF13A1TGM2TGM1
SCHEMBL31634669 0.83 RORC (0.35) GRIN2BF13A1TGM2TGM1NPC1
SCHEMBL30948971 0.83 RORC (0.35) GRIN2BF13A1TGM2TGM1NPC1
SCHEMBL30948983 0.82 PTGDR2 (0.35) GRIN2BKDM1AF13A1TGM2TGM1
SCHEMBL31634678 0.82 PTGDR2 (0.35) GRIN2BKDM1AF13A1TGM2TGM1
SCHEMBL30948981 0.79 RAB9A (0.44) GRIN2BF13A1TGM2TGM1NPC1
SCHEMBL31634718 0.79 RAB9A (0.44) GRIN2BF13A1TGM2TGM1NPC1
SCHEMBL30948974 0.76 GRM5 (0.44) GRIN2BF13A1TGM2TGM1NPC1
SCHEMBL31634701 0.76 GRM5 (0.44) GRIN2BF13A1TGM2TGM1NPC1
SCHEMBL30948984 0.74 NR1H2 (0.46) GRIN2BF13A1TGM2TGM1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024104452-A1 MC4R ANTAGONIST COMPOUND, PHARMACEUTICAL COMPOSITION AND PHARMACEUTICAL USE THEREOF 长春金赛药业有限责任公司 2024-05-23 WO disclosed