SCHEMBL30948971

SCHEMBL30948971

Cc1nc(N[C@@H]2CN(C(=O)OCc3ccccc3)CC23CC3)ccc1-c1cn(C)c(C(C)(C)O)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.35
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
MC4R P32245 2/20 0.33
KCNH2 Q12809 1/20 0.33
F13A1 P00488 1/20 0.33
TGM2 P21980 1/20 0.33
TGM1 P22735 1/20 0.33
CCR5 P51681 1/20 0.33
CHRM4 P08173 1/20 0.33
HTT P42858 1/20 0.33
ENPP2 Q13822 4/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PARP1 P09874 1/20 0.32
ACACB O00763 1/20 0.32
ATXN2 Q99700 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31634669 1.00 RORC (0.35) RORCPDK1PDK2PDK3PDK4
SCHEMBL31634678 0.85 PTGDR2 (0.35) RORCF13A1TGM2TGM1CCR5
SCHEMBL30948983 0.85 PTGDR2 (0.35) RORCF13A1TGM2TGM1CCR5
SCHEMBL31634667 0.83 GRIN2B (0.36) RORCF13A1TGM2TGM1ENPP2
SCHEMBL30948965 0.83 GRIN2B (0.36) RORCF13A1TGM2TGM1ENPP2
SCHEMBL31634718 0.80 RAB9A (0.44) RORCF13A1TGM2TGM1CHRM4
SCHEMBL30948981 0.80 RAB9A (0.44) RORCF13A1TGM2TGM1CHRM4
SCHEMBL31634688 0.78 PIM1 (0.32) MC4RKCNH2F13A1TGM2TGM1
SCHEMBL31634701 0.77 GRM5 (0.44) RORCF13A1TGM2TGM1HTT
SCHEMBL30948974 0.77 GRM5 (0.44) RORCF13A1TGM2TGM1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024104452-A1 MC4R ANTAGONIST COMPOUND, PHARMACEUTICAL COMPOSITION AND PHARMACEUTICAL USE THEREOF 长春金赛药业有限责任公司 2024-05-23 WO disclosed